EC Number | Crystallization (Comment) | Organism |
---|---|---|
3.4.21.21 | hanging drop vapour diffusion method | Homo sapiens |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.21.21 | R-4-[2-(3-aminobenzenesulfonylamino)-1-(3,5-diethoxy-2-fluorophenyl)-2-oxoethylamino]-2-hydroxy-benzamidine | incubation with enzyme in 100 mM Hepes, pH 7.8, 140 mM NaCl, 0.1% (v/v) polyethylene glycol 8000, 0.02% (v/v) Tween 80, 5 mM CaCl2 for 40 min at room temperature | Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.21.21 | Homo sapiens | P08709 | - |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.21.21 | factor X + H2O | - |
Homo sapiens | factor Xa | - |
? | |
3.4.21.21 | N-methylsulfonyl-D-phenyl-D-glycyl-D-arginyl-4-nitroanilide + H2O | - |
Homo sapiens | N-methylsulfonyl-D-phenyl-D-glycyl-D-arginine + 4-nitroaniline | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.21.21 | FVIIa | - |
Homo sapiens |
3.4.21.21 | serine protease factor VIIa | - |
Homo sapiens |
3.4.21.21 | TF-FVIIa | factor VIIa in complex with tissue factor | Homo sapiens |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.21.21 | 0.00000035 | - |
R-4-[2-(3-aminobenzenesulfonylamino)-1-(3,5-diethoxy-2-fluorophenyl)-2-oxoethylamino]-2-hydroxy-benzamidine | - |
Homo sapiens |